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Ampasse is a Russian intravenous nootropic, the calcium salt of 5-hydroxynicotinoyl glutamate, presented as an ampakine that modulates AMPA type glutamate receptors in chronic cerebrovascular disease.
- Intravenous nootropic used in chronic cerebrovascular disease
- Glutamate coupled to hydroxylated nicotinic acid
- Presented as an ampakine at AMPA type receptors
- Same carrier trick picamilon uses
- Rare Russian pharmacology, seldom seen outside one country
Mechanism
Structurally it is coupled to a hydroxylated acid, the same design idea as picamilon, which couples nicotinic acid to to carry it across the blood brain barrier. The manufacturer describes positive modulation of subtype glutamate receptors along with antidepressant, anxiolytic and neuroprotective activity. No independent binding or electrophysiology work confirms an ampakine action, so calling it one is at present the developer's claim rather than a replicated finding, and the entry should say so rather than repeat the classification.
Safetyrisks and cautions, not medical advice
an intravenous-only prescription drug registered in Russia alone, whose entire clinical and mechanistic record comes from the developer's own programme
Subjective profileweighing the evidence above
Calling this an ampakine is the developer's description rather than a replicated finding, and that distinction is the entire entry. No independent binding or electrophysiology work confirms positive AMPA modulation, the clinical record comes from the programme that owns the molecule, and registration exists in one country. The structural idea is not silly, since coupling nicotinic acid to a neurotransmitter is the same trick picamilon uses, but a plausible structure is not evidence of an effect. Intravenous administration settles the rest: this is a hospital product, not something a reader can evaluate or obtain sensibly.
Where to buy
Suppliers
Vendors carrying Ampasse, with live product details and codes. Links are affiliate links that support the wiki at no cost to you.
RUPharma🌐
Ampasse