Loading…
for educational and safety purposes
class, effects, and the receptor fingerprint, side by side; add up to four, then source the whole stack
Popular head-to-heads →alpha-2-delta-1 calcium channel subunitbinds
Neuropathic pain signalingdampens
Nervous system excitabilitylowers
a2d-1 subunit of voltage-gated Ca2+ channels (CACNA2D1)Binds / inhibits (via active gabapentin)
a2d-2 subunit of voltage-gated Ca2+ channels (CACNA2D2)Binds
MCT-1 transporter (SLC16A1)Substrate (absorption)
SMVT transporter (SLC5A6)Substrate (absorption)
GABA-A / GABA-B receptorsNo direct binding
checking Gabapentin and Gabapentin enacarbil: no notable interaction flagged; they read as broadly independent.
no notable interaction flagged; these look broadly independent.
General educational info, not medical advice.